JTP-117968
JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation.
For research use only. We do not sell to patients.
- CAS No.: 2250132-99-9
- Formula: C31H31F3N2O2
- Molecular Weight:520.59
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2250132-99-9
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Molecular Weight 520.59
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Formula C31H31F3N2O2
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SMILES
O=C(C(C=C1C2)=CC=C1[C@]3(CC4=CC=CC=C4)CC[C@@](C(F)(F)F)(O)C[C@@]3([H])C52CC5)NC6=CC=CN=C6C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)