1. GPCR/G Protein
  2. Glucocorticoid Receptor
  3. JTP-117968

JTP-117968 

Cat. No.: HY-125265
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JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation.

For research use only. We do not sell to patients.

JTP-117968 Chemical Structure

JTP-117968 Chemical Structure

CAS No. : 2250132-99-9

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Description

JTP-117968, a novel selective glucocorticoid receptor modulator (a non-steroidal SGRM, IC50 of 6.8 nM), exhibits improved transrepression/transactivation dissociation[1].

In Vitro

JTP-117968 has partial TR activity, but exhibits extremely low TA activity[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

520.59

Formula

C31H31F3N2O2

CAS No.
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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
JTP-117968
Cat. No.:
HY-125265
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