PF-622
Based on 1 publication(s) in Google Scholar
PF-622 is a selective FAAH inhibitor, and can be used for study of analgesic and anxiolytic/antidepressant.
연구목적의 판매만을 진행합니다. 환자를 대상으로 한 판매는 하지 않습니다.
- CAS No.: 898235-65-9
- 화학식: C21H22N4O
- 분자량:346.43
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보관:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
Publications Citing Use of MedChemExpress (MCE) PF-622
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Biological Activity
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HEK293 | EC50 |
>25 μM
Compound: PF-622
|
Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as decrease in intracellular calcium level
Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as decrease in intracellular calcium level
|
[PMID: 19875281] |
| HEK293 | IC50 |
>10 μM
Compound: PF-622
|
Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium level
Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as decrease in intracellular calcium level
|
[PMID: 19875281] |
Chemical Information
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CAS No. 898235-65-9
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Appearance Solid
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분자량 346.43
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화학식 C21H22N4O
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SMILES
O=C(N1CCN(CC1)CC2=NC3=C(C=C2)C=CC=C3)NC4=CC=CC=C4
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
Publications (1)
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Journal Impact Factor
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Most Recent
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Chin Med
Electroacupuncture to point Baihui confers anxiolytic effects by promoting oxytocin release from PVN in Mice. [Abstract]2026 Jan 13;21(1):30. PMID: 41530867
순도&문서
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)