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Cat. No.: HY-123142

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RX809055AX

RX 809055AX is a potent long lasting opioid antagonist with selectivity towards at mu and delta receptors.

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CAS No.: 122566-12-5
화학식: C₂₉H₂₉ClN₂O₄
분자량:505.00

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (275 KB)

RX809055AX Chemical Structure

CAS No.: 122566-12-5

Amount: USD 0.00

* 장바구니에 담기 전 물품의 수량을 선택해 주십시오.

Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity
- 제품 설명
- IC₅₀ & Target
- Cellular Effect
Chemical Information
순도&문서
References
Calculators
Help & FAQs
Classifications
Bioz

Biological Activity

제품 설명

RX 809055AX is a potent long lasting opioid antagonist with selectivity towards at mu and delta receptors^[1].

IC₅₀ & Target

μ Opioid Receptor/MOR

δ Opioid Receptor/DOR

All Opioid Receptor Isoforms :

Cellular Effect

Cell Line	Type	Value	Description	References
CHO	IC₅₀	0.1 nM Compound: 4a, C-CAM	Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant kappa opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]
CHO	IC₅₀	0.19 nM Compound: 4a, C-CAM	Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant delta opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]
CHO	IC₅₀	0.53 nM Compound: 4a, C-CAM	Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding Activity at human recombinant mu opioid receptor expressed in CHO cells assessed as stimulation of [35S]GTP-gamma-S binding	[PMID: 17004724]

Chemical Information

CAS No. 122566-12-5
분자량 505.00
화학식 C₂₉H₂₉ClN₂O₄
SMILES

ClC(C=C1)=CC=C1/C=C/C(N[C@]23[C@@]45C6=C(C[C@@]3([H])N(CC5)CC7CC7)C=CC(O)=C6O[C@@]4([H])C(CC2)=O)=O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (275 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Lemcke PK, Ayres EA, Kramer TH, Burks TF. RX809055AX in vivo: a long lasting opioid antagonist at mu and delta receptors. Proc West Pharmacol Soc. 1989;32:173-5. [Content Brief]

Calculators

몰농도 계산기

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

농도 희석 계산기

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

Bioz

Keywords

MOQ

Minimum order quantity

100 mg

견적 받기 해외재고보유

Other size

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Amount: USD 0.00

Biological Activity
- 제품 설명
- IC₅₀ & Target
Chemical Information
순도&문서
References

상품명:
Cat. No.:
수량:
MCE Japan Authorized Agent:

상품명:
CAS No.:
Species:
Purity:
수량:

RX809055AX

All Opioid Receptor Isoforms

Biological Activity

제품 설명

IC50 & Target

Cellular Effect

Chemical Information

순도&문서

References

Calculators

Help & FAQs

RX809055AX Related Classifications

HY-123142 Related Classifications

Bioz

Keywords

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