1. GPCR/G Protein
    Neuronal Signaling
  2. MCHR1 (GPR24)
  3. MCHR1 antagonist 3

MCHR1 antagonist 3 

Cat. No.: HY-136152
Handling Instructions

MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism.

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MCHR1 antagonist 3 Chemical Structure

MCHR1 antagonist 3 Chemical Structure

CAS No. : 1069622-60-1

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Description

MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].

In Vitro

Compound 1, derived from a spirohydantoin scaffold, exhibits a Ki of 50 nM at MCH-R1. Compound 1 is a potent inhibitor of CYP3A4 (IC50=35 nM). MCHR1 antagonist 3 is an analog of compound 1[1].

Molecular Weight

472.62

Formula

C₂₉H₃₆N₄O₂

CAS No.

1069622-60-1

SMILES

O=C(N1C2CC3=C(C=CC=C3)C2)N(CC)C4(CCN(CC5=CC=C(N6CCCC6)C=C5)CC4)C1=O

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Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Keywords:

MCHR1 antagonist 3MCHR1 (GPR24)Melanin concentrating hormone receptor 1melanin-concentratinghormonereceptor-1energymetabolismInhibitorinhibitorinhibit

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MCHR1 antagonist 3
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