Metrenperone
Metrenperone is an inhibitor for 5-HT2 receptor. Metrenperone exhibits α1 and α2 antagonist activity as well as anti-H1 and anti-dopaminergic efficacy. Metrenperone can lower the blood pressure, enhances bradycardia in peripheral ischemia, inhibits serotonin-induced platelet aggregation, and antagonizes serotonin-mediated vasoconstriction. Metrenperone promotes the repair of acutely damaged collagen tissue.
For research use only. We do not sell to patients.
- CAS No.: 81043-56-3
- Formula: C24H26FN3O2
- Molecular Weight:407.48
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All Adrenergic Receptor Isoforms
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Biological Activity
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α1-adrenergic receptor |
α2-adrenergic receptor |
Chemical Information
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CAS No. 81043-56-3
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Molecular Weight 407.48
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Formula C24H26FN3O2
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SMILES
O=C1C(CCN2CCC(CC2)C(C3=CC=C(C=C3)F)=O)=C(N=C4N1C=C(C=C4)C)C
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
[1]. Oryan A, et al., Effects of a serotonin S2-receptor blocker on healing of acute and chronic tendon injuries. J Invest Surg. 2009 Jul-Aug;22(4):246-55. [Content Brief]
[2]. Linden A, et al., Cardiovascular response to intravenous administration of 5-hydroxytryptamine after type-2 receptor blockade, by metrenperone, in healthy calves. Vet J. 1999 Jan;157(1):31-7. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Metrenperone Related Classifications
HY-121311 Related Classifications
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