MRGPRX4 modulator-3
MRGPRX4 modulator-3 (Compound 1C) is a negative allosteric MAS-related G-protein-coupled receptor X4 (MRGPRX4) modulator. MRGPRX4 modulator-3 significantly attenuates Nateglinide (HY-B0422) (orthosteric agonist)-induced responses with an IC50 of 337 nM. MRGPRX4 modulator-3 can be used for chronic itch (especially cholestatic itch) and pain research.
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- No. CAS: 3137192-95-8
- Fòrmula: C19H22FN3S
- Peso molecular:343.46
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Almacenamiento:
Please store the product under the recommended conditions in the Certificate of Analysis.
Actividad biológica
Descripciòn
Chemical Information
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No. CAS 3137192-95-8
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Peso molecular 343.46
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Fòrmula C19H22FN3S
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SMILES
C[C@]1(C2(C)C)/C(C[C@@H]2CC1)=N\NC3=NC(C4=CC=C(F)C=C4)=CS3
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Envío
Room temperature in continental US; may vary elsewhere.
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Almacenamiento
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureza y Documentación
Referencias
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)