P2X3 antagonist 38
P2X3 antagonist 38 (compound 4) is a potent and orally active P2X3 antagonist with IC50 values of 0.132, 0.165, 0.421 µM for hP2X3, rP2X3, gpP2X3, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2545974-71-6
- Formula: C22H25F3N6O3
- Molecular Weight:478.47
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All P2X Receptor Isoforms
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Biological Activity
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P2X3 Receptor 0.132 μM (IC50) |
Chemical Information
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CAS No. 2545974-71-6
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Molecular Weight 478.47
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Formula C22H25F3N6O3
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SMILES
CCOC(N([C@@H]1C(C2=CC=C(C=C2)C)=NN(C1)C(N[C@@H](C3=CN=C(C(F)(F)F)N=C3)C)=O)C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)