2. Others GPCR/G Protein
  3. Drug Derivative Bombesin Receptor
  4. PD 168368 derivative-1

PD 168368 derivative-1 (Compound 16) is a derivative of PD 168368 (HY-116216), with Ki values of 0.46 and 3.7 nM for the subtypes of bombesin receptor (BB₁ and BB₂). PD 168368 derivative-1 can be used for the study of various diseases, such as cancer, depression, and eating disorders.

For research use only. We do not sell to patients.

PD 168368 derivative-1

PD 168368 derivative-1 Chemical Structure

CAS No. : 216319-58-3

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PD 168368 derivative-1 Related Antibodies

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Description

PD 168368 derivative-1 (Compound 16) is a derivative of PD 168368 (HY-116216), with Ki values of 0.46 and 3.7 nM for the subtypes of bombesin receptor (BB₁ and BB₂). PD 168368 derivative-1 can be used for the study of various diseases, such as cancer, depression, and eating disorders[1].

Molecular Weight

583.68

Formula

C33H37N5O5
CAS No.
SMILES

O=N(C(C=C1)=CC=C1NC(N[C@](CC2=CNC3=CC=CC=C23)(C)C(NCC4(C5=CC=C(C=C5)OC)CCCCC4)=O)=O)=O
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Room temperature in continental US; may vary elsewhere.
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Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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PD 168368 derivative-1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

PD 168368 derivative-1216319-58-3Drug DerivativeBombesin ReceptorDrug derivativeBombesinBB1 receptorBB2 receptornon-peptide antagonistPD 176252structure-activity relationshipInhibitorinhibitorinhibit

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PD 168368 derivative-1
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HY-17673
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