(R)-(-)-α-Methylhistamine
For research use only. We do not sell to patients.
- CAS No.: 75614-87-8
- Formula: C6H11N3
- Molecular Weight:125.17
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Cellular Effect
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| CHO | EC50 |
2.8 nM
Compound: 1
|
Agonist activity at human recombinant histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintillation counting
Agonist activity at human recombinant histamine H3 receptor expressed in CHO cells assessed as [35S]GTPgammaS binding after 1 hr by liquid scintillation counting
|
[PMID: 20384344] |
| CHO-K1 | IC50 |
2.3 nM
Compound: RAMH
|
Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHOK1 cells after 2 hrs
Displacement of [3H]N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHOK1 cells after 2 hrs
|
[PMID: 23403082] |
Chemical Information
-
CAS No. 75614-87-8
-
Molecular Weight 125.17
-
Formula C6H11N3
-
SMILES
C[C@@H](N)CC1=CN=CN1
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Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)