Riodipine
Riodipine (PP-1466) is a vasodilator. Riodipine can be used for the research of antihypertensive.
Nur für Forschungszwecke. Wir verkaufen nicht an Patienten.
- CAS. Nr.: 71653-63-9
- Formel: C18H19F2NO5
- Molecular Weight:367.34
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Speicherung:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biologische Aktivität
Riodipine;Foridon;PP 1466;PP1466;PP-1466
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| HepG2 | EC50 |
1.6 μM
Compound: Riodipine
|
Activation of human PXR expressed in human HepG2 (DPX-2) cells assessed as induction of CYP3A4 after 24 hrs by luminescent analysis
Activation of human PXR expressed in human HepG2 (DPX-2) cells assessed as induction of CYP3A4 after 24 hrs by luminescent analysis
|
[PMID: 20966043] |
| HepG2 | EC50 |
1.8 μM
Compound: Riodipine
|
Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysis
Activation of rat PXR expressed in human HepG2 cells after 24 hrs by luciferase reporter gene based luminescent analysis
|
[PMID: 20966043] |
| HepG2 | EC50 |
4 μM
Compound: Riodipine
|
Activation of human PXR expressed in human HepG2 (DPX-2) cells after 24 hrs by luciferase reporter gene based luminescent analysis
Activation of human PXR expressed in human HepG2 (DPX-2) cells after 24 hrs by luciferase reporter gene based luminescent analysis
|
[PMID: 20966043] |
Chemical Information
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CAS. Nr. 71653-63-9
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Molecular Weight 367.34
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Formel C18H19F2NO5
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SMILES
O=C(OC)C1=C(NC(C)=C(C1C2=CC=CC=C2OC(F)F)C(OC)=O)C
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Synonyms
Foridon; PP-1466
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Versand
Room temperature in continental US; may vary elsewhere.
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Speicherung
Please store the product under the recommended conditions in the Certificate of Analysis.
Reinheit & Dokumentation
Verweise
Calculators
Konzentration (Stammlösung) × Volumen (Stammlösung) = Konzentration (Ziellösung) × Volumen (Ziellösung)