59 Results for "

B2+receptor

" in MedChemExpress (MCE) Product Catalog:
Products (59)

59 Results for "B2+receptor" in MCE Product Catalog:

Cat. No.: HY-P2118
CAS No.: 109333-26-8
Target:  

Bradykinin Receptor

Research Areas:  

Inflammation/Immunology

NPC-567 is a bradykinin B2 receptor antagonist. NPC-567 is effective in inhibiting the acute response to allergen in the airways [2].
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Cat. No.: HY-123376
CAS No.: 193344-25-1
Target:  

Bradykinin Receptor

Research Areas:  

Neurological Disease

FR-190997 is a non-peptide Bradykinin B2 receptor selective agonist, Ki value is 9.8 nM. FR-190997 is also an effective antihypertensive agent .
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Cat. No.: HY-14886
CAS No.: 1157852-02-2
Synonyms: MEN16132 free base
Fasitibant chloride (MEN16132 free base) is a potent and selective nonpeptide bradykinin B2 receptor (B2R) antagonist. Fasitibant chloride reduces joint pain and diminishes joint oedema in Carrageenan-induced arthritis rat model [2] .
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Cat. No.: HY-100301
CAS No.: 215258-13-2
FR167344 free base is an orally active, nonpeptide bradykinin receptor B2 antagonist. FR167344 free base shows a high affinity binding to the B2 receptor with an IC50 value of 65 nM and no binding affinity for the B1 receptor.
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Cat. No.: HY-118945
CAS No.: 194928-55-7
FR191413 is a selective bradykinin B2 receptor agonist that stimulates prostaglandin E2 production in WI-38 cells and activates BK B2 receptor-mediated pathways such as vasodilation and organ protection. FR191413 competitively binds to [ 3H]-BK in guinea pig ileum (GPI) membranes and CHO cells transfected with the human BK B2 receptor, with IC50 values ​​of 20.0 nM and 2.60 nM, respectively. FR191413 can be used in research related to cardiovascular diseases and diabetes, including hypertension, myocardial hypertrophy, myocardial infarction, arrhythmias, and diabetic nephropathy .
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Cat. No.: HY-P5493
CAS No.: 103412-42-6
Target:  

Inhibitory Antibodies

Research Areas:  

Others

D-Arg-[Hyp3,Thi5,8,D-Phe7]-Bradykinin is a biological active peptide. (inhibited bradykinin-induced contractions concentration dependently; bradykinin B2 receptor antagonist)
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Cat. No.: HY-103294
CAS No.: 229030-05-1
Target:  

Endogenous Metabolite

Research Areas:  

Others

R892 is a selective and efficient bradyKinin B1 receptor antagonist with significant antagonistic activity. The pA2 values of R892 in human and rabbit B1 receptors are 8.8 and 8.6 respectively, indicating its strong anti-activity at these receptors. R892 exhibits selectivity with ID50 values of 2.8 nM and >600 nM for B1 and B2 receptors, respectively, and has no endogenous agonist activity. R892 is resistant to aminopeptidase and kininase II (ACE) degradation and exhibits metabolic stability .
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Cat. No.: HY-P1650
CAS No.: 215713-39-6
Synonyms: B 9870
Target:  

Bradykinin Receptor ERK

Research Areas:  

Cancer

Breceptin (B 9870) is an antagonist of the bradykinin B1/B2 receptor (B1/B2R). Breceptin exhibits an irreversible antagonist effect on B2R, inhibiting the vasodilation induced by Bradykinin (HY-P0206) in the rabbit carotid vein contraction experiment. B-9870 shows partial agonist properties in HEK 293 cells with high expression of B2R, and can activate ERK1/2 phosphorylation, calcium ion mobilization, arachidonic acid release, and receptor internalization. Breceptin can be used in research to inhibit breast cancer and non-small cell lung cancer .
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Cat. No.: HY-P70841
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P73035
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P73037
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Rat
Source:  
HEK293
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Cat. No.: HY-P700733
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P705611
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Mouse
Source:  
HEK293
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Cat. No.: HY-P73036
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Rat
Source:  
HEK293
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Cat. No.: HY-P78454
Purity:  ≥ 95%, as determined by Bis-Tris PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P701234
Purity:  ≥ 95%, as determined by Bis-Tris PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-P702752
Purity:  ≥ 70%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human
Source:  
Sf9 insect cells
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Cat. No.: HY-P703899
Purity:  ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: ERBB4; Proto-Oncogene-Like Protein C-ErbB-4; Erb-B2 Receptor Tyrosine Kinase 4; P180erbB4; HER4; V-Erb-A Avian Erythroblastic Leukemia Viral Oncogene Homolog-Like 4; ALS19; Avian Erythroblastic Leukemia Viral (V-Erb-B2) Oncogene Homolog 4; V-Erb-B2 Avian
Species:  
Human Rhesus Macaque
Source:  
HEK293
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Cat. No.: HY-P73000
Purity:  ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: EPHB2; Ephrin Type-B Receptor 2 Variant; Prev. EPHT3; Protein-Tyrosine Kinase HEK5; Prev. DRT; Elk-Related Tyrosine Kinase; Prev. ERK; ELK-Related Tyrosine Kinase; Tyrosine-Protein Kinase Receptor EPH-3; Eph Tyrosine Kinase 3; Ephrin Type-B Receptor 2; EPH Tyrosine Kinase 3; Tyro5; BDPLT22; Hek5; EphB2; Developmentally-Regulated Eph-Related Tyrosine Kinase; TYRO5; Renal Carcinoma Antigen NY-REN-47; EPTH3; Tyrosine-Protein Kinase TYRO5; CAPB; EPH-Like Kinase 5; PCBC; EK5; HEK5; EPH Receptor B2; Receptor Protein-Tyrosine Kinase
Species:  
Human
Source:  
Sf9 insect cells
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Cat. No.: HY-P70857
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: ERBB3; Receptor Protein-Tyrosine Kinase; Prev. LCCS2; P45-SErbB3; HER3; P85-SErbB3; V-Erb-B2 Avian Erythroblastic Leukemia Viral Oncogene Homolog 3; ErbB-3 R31; Tyrosine Kinase-Type Cell Surface Receptor HER3; MDA-BF-1; Human Epidermal Growth Factor Receptor 3; C-ErbB3; Receptor Tyrosine-Protein Kinase ErbB-3; ErbB3-S; Proto-Oncogene-Like Protein C-ErbB-3; ErbB-3; C-ErbB-3; FERLK; CDNA FLJ43038 Fis, Clone BRTHA3002955, Highly Similar To Receptor Tyrosine-Protein Kinase ErbB-3; VSCN1; Lethal Congenital Contracture Syndrome 2; Erb-B2 Receptor Tyrosine Kinase 3; P180-ErbB3
Species:  
Mouse
Source:  
HEK293
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