3 Results for "

ARC239

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "ARC239" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-12709
CAS No.: 67339-62-2
Purity:  99.71%
Research Areas:  

Neurological Disease

ARC 239 is an α2B/C-adrenergic receptor antagonist with pKi of 7.06 and 6.95 for rat kidney α2B and human α2C, respectively. ARC 239 also inhibits 5-HT1A receptor with a Ki of 63.1 nM .
loading...
    loading...
2
2 Cited Publications
Cat. No.: HY-12709A
CAS No.: 55974-42-0
Purity:  99.57%
ARC 239 dihydrochloride is a selective α2B/2C adrenoceptor antagonist (pKd values are 5.95, 7.41 and 7.56 at α2A, α2B, and α2C receptors respectively). ARC 239 dihydrochloride binds to CHO cell membranes expressing human recombinant a2A-, a2B- or a2C-adrenoceptor subtypes with pKis of 5.6, 8.4, and 7.08, respectively .
loading...
    loading...
Cat. No.: HY-12709R
CAS No.: 67339-62-2
Research Areas:  

Neurological Disease

ARC 239 (Standard) is the analytical standard of ARC 239. This product is intended for research and analytical applications. ARC 239 is an α2B/C-adrenergic receptor antagonist with pKi of 7.06 and 6.95 for rat kidney α2B and human α2C, respectively. ARC 239 also inhibits 5-HT1A receptor with a Ki of 63.1 nM .
loading...
    loading...