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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
2 Results for "
Azapetine
" in MedChemExpress (MCE) Product Catalog:
Products (2)
2 Results for "Azapetine" in MCE Product Catalog:
Target:
Research Areas:
Azapetine is an α-adrenergic receptor antagonist, with a IC50 of 0.205 μM against rat α1-adrenergic receptors and a IC50 of 1.3 μM against rat α2-adrenergic receptors. Azapetine blocks α1/α2-adrenergic receptor-mediated contraction of blood vessels and vascular smooth muscles. Azapetine can be used for the research of peripheral vascular diseases .
Cat. No.: HY-W745352
CAS No.: 65-15-6
Target:
Research Areas:
Azapetine hydrochloride is a selective α1-adrenergic receptor inhibitor with an IC50 of 205 nM. Azapetine hydrochloride inhibits Epinephrine (HY-B0447)-induced platelet aggregation, slightly enhances the contractile response of isolated rat vas deferens, and blocks α1 and α2 adrenergic receptor-mediated vasoconstriction .
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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
