1 Result for "

BDCM

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "BDCM" in MCE Product Catalog:

Cat. No.: HY-155245
CAS No.: 2911646-14-3
Target:  

CDK Bcl-2 Family

Research Areas:  

Cancer

A09-003 is a CDK-9 inhibitor (IC50: 16 nM). A09-003 inhibits leukemia cell proliferation (IC50: 1.90, 0.86, 2.49, 1.84, 0.48 μM for BDCM, Molm-14, THP-1, U937, MV4-11 cells). A09-003 induces apoptosis and decreases Mcl-1 expression through Thr163 dephosphorylation .
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