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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
10 Results for "
GPR91
" in MedChemExpress (MCE) Product Catalog:
Products (10)
10 Results for "GPR91" in MCE Product Catalog:
14
14 Publications Verification
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Research Areas:
NF-56-EJ40 is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM .
14
14 Publications Verification
Cat. No.: HY-130246A
CAS No.: 2728500-80-7
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NF-56-EJ40 hydrochloride is a potent, high-affinity, and highly selective human SUCNR1 (GPR91) antagonist with an IC50 of 25 nM and a Ki of 33 nM, and shows almost no activity towards rat SUCNR1. NF-56-EJ40 hydrochloride has high affinity for humanized rat SUCNR1 with a Ki value of 17.4 nM .
3
3 Cited Publications
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hGPR91 antagonist 1 (Compound 4c) is a potent and selective GPR91 antagonist with an IC50 of 7 nM for human GPR91 .
3
3 Cited Publications
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cis-Epoxysuccinic acid is a succinate receptor (SUCNR1/GPR91) agonist. cis-Epoxysuccinic acid inhibits cAMP levels with an EC50 value of 2.7 μM. cis-Epoxysuccinic acid can be used for the research of cardiovascular system .
1
1 Cited Publications
Cat. No.: HY-RS14004
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Sucnr1 Mouse Pre-designed siRNA Set A contains three designed siRNAs for Sucnr1 gene (Mouse), as well as a negative control, a positive control, and a FAM-labeled negative control.
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hGPR91 antagonist 3 (Compound 5g) is a potent and orally active GPR91 antagonist with IC50s of 35 nM and 135 nM, for human GPR91 and rat GPR91, respectively .
Cat. No.: HY-RS14003
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SUCNR1 Human Pre-designed siRNA Set A contains three designed siRNAs for SUCNR1 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.
Cat. No.: HY-W693142
CAS No.: 140-99-8
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Research Areas:
Succinate calcium is a key intermediate product of the citric acid cycle (tricarboxylic acid cycle). Succinate calcium can act as a specific ligand for the G protein-coupled receptor GPR91. Succinate calcium can increase the amplitude of calcium transient in cardiac muscle cells and accelerate the decay rate of calcium transient. Succinate calcium can induce myocardial apoptosis .
Cat. No.: HY-P705683
Purity: ≥ 85%, as determined by reducing SDS-PAGE.
Synonyms: Succinate receptor 1 Curated; Alternative names; G-protein coupled receptor 91; P2Y purinoceptor 1-like; SUCNR1; GPR91
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Cat. No.: HY-RS14005
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Sucnr1 Rat Pre-designed siRNA Set A contains three designed siRNAs for Sucnr1 gene (Rat), as well as a negative control, a positive control, and a FAM-labeled negative control.
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
