7 Results for "

Lys76

" in MedChemExpress (MCE) Product Catalog:
Products (7)

7 Results for "Lys76" in MCE Product Catalog:

3
3 Cited Publications
Cat. No.: HY-P0227
CAS No.: 168482-23-3
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

SHU 9119 is a potent human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist; with IC50 values of 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively.
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1
1 Cited Publications
Cat. No.: HY-18678A
CAS No.: 1607799-13-2
Synonyms: PT-141 Acetate
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

Bremelanotide (PT-141) Acetate is a melanocortin receptor agonist. Bremelanotide Acetate can activate MC4R and increases dopamine release. Bremelanotide Acetate induces appetitive sexual behaviors, female mounting behavior, and repetitive self-grooming. Bremelanotide Acetate can be used for the research of hypoactive sexual desire disorders .
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Cat. No.: HY-121629
CAS No.: 1221962-86-2
Purity:  98.02%
Target:  

PDK-1

Research Areas:  

Cancer

PS210 is a potent and selective PDK1 activator with a Kd of 3 μM and targets the PIF-binding pocket of PDK1. PS210 is inactive against other protein kinases, including PDK1 downstream signaling components such as S6K, PKB/Akt or GSK3. In cells, the prodrug of PS210 (PS423) acts as a substrate-selective inhibitor of PDK1, inhibiting the phosphorylation and activation of S6K .
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Cat. No.: HY-P1208
CAS No.: 667430-81-1
Target:  

Melanocortin Receptor

Research Areas:  

Inflammation/Immunology

PG-931, an analog of SHU 9119 (HY-P0227), is a potent melanocortin 4 (MC4) receptor (IC50=0.58 nM) agonist and is more selective than for the hMC3R (IC50=55 nM) or the hMC5R (IC50=2.4 nM). PG-931 can reverse haemorrhagic shock and prevent multiple organ damage in vivo .
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Cat. No.: HY-P1209A
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

PG106 TFA is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50= 210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor .
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Cat. No.: HY-P1209
CAS No.: 944111-22-2
Target:  

Melanocortin Receptor

Research Areas:  

Inflammation/Immunology

PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor .
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Cat. No.: HY-P1208A
Target:  

Melanocortin Receptor

Research Areas:  

Inflammation/Immunology

PG-931 TFA, an analog of SHU 9119 (HY-P0227), is a potent melanocortin 4 (MC4) receptor (IC50=0.58 nM) agonist and is more selective than for the hMC3R (IC50=55 nM) or the hMC5R(IC50=2.4 nM). PG-931 TFA can reverse haemorrhagic shock and prevent multiple organ damage in vivo .
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