1. GPCR/G Protein
    Neuronal Signaling
  2. Melanocortin Receptor
  3. PG106

PG106 

Cat. No.: HY-P1209
Handling Instructions

PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor.

For research use only. We do not sell to patients.

Custom Peptide Synthesis

PG106 Chemical Structure

PG106 Chemical Structure

CAS No. : 944111-22-2

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Description

PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor[1].

IC50 & Target

IC50: 210 nM (hMC3 receptor)
EC50: 9900 nM (hMC4 receptor)[1]

Molecular Weight

1008.18

Formula

C₅₁H₆₉N₁₃O₉

CAS No.

944111-22-2

Sequence Shortening

Ac-{Nle}-D-{Bal}-{D-Nal}-RWK-NH2 (Lactam bridge:Asp2-Lys7)

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

References
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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

PG106PG 106PG-106Melanocortin ReceptorMC ReceptormelanocortinhMC3hMC4hMC5lactam derivativeInhibitorinhibitorinhibit

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PG106
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HY-P1209
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