PG106
PG106 is a potent and selective human melanocortin 3 (hMC3) receptor antagonist (IC50=210 nM) and has noactivity at hMC4 receptors (EC50=9900 nM) and hMC5 receptor.
For research use only. We do not sell to patients.
- CAS No.: 944111-22-2
- Formula: C51H69N13O9
- Molecular Weight:1008.18
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 210 nM (hMC3 receptor)EC50: 9900 nM (hMC4 receptor)[1]
Chemical Information
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CAS No. 944111-22-2
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Molecular Weight 1008.18
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Formula C51H69N13O9
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Sequence Shortening
Ac-{Nle}-D-{Bal}-{D-Nal}-RWK-NH2 (Lactam bridge:Asp2-Lys7)
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)