6 Results for "

Methiothepin

" in MedChemExpress (MCE) Product Catalog:
Products (6)

6 Results for "Methiothepin" in MCE Product Catalog:

Cat. No.: HY-111491
CAS No.: 20229-30-5
Synonyms: Metitepine; Ro 8-6837
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Methiothepin (Metitepine; Ro 8-6837) is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
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2
2 Cited Publications
Cat. No.: HY-107836
CAS No.: 74611-28-2
Purity:  99.60%
Synonyms: Metitepine mesylate; Ro 8-6837 mesylate
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Methiothepin (Metitepine) mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
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Cat. No.: HY-101009
CAS No.: 19728-88-2
Synonyms: Metitepine maleate; Ro-8-6837 maleate
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Methiothepin maleate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
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Cat. No.: HY-107836R
CAS No.: 74611-28-2
Synonyms: Metitepine mesylate (Standard); Ro 8-6837 mesylate (Standard)
Research Areas:  

Neurological Disease

Methiothepin (mesylate) (Standard) is the analytical standard of Methiothepin (mesylate). This product is intended for research and analytical applications. Methiothepin (Metitepine) mesylate is a potent and non-selective 5-HT2 receptor antagonist, with pKds of 7.10 (5-HT1A), 7.28 (5HT1B), 7.56 (5HT1C), 6.99 (5HT1D), 7.0 (5-HT5A), 7.8 (5-HT5B), 8.74 (5-HT6), and 8.99 (5-HT7), and pKis of 8.50 (5HT2A), 8.68 (5HT2B), and 8.35 (5HT2C).
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Cat. No.: HY-P12260
CAS No.: 3027489-02-4
Research Areas:  

Cancer

AJICAP reagent 1b is a thiophenyl ester-based site-specific conjugation reagent for antibody modification applications. AJICAP reagent 1b is used in HER2-positive gastric cancer-related research .
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Cat. No.: HY-P12261
Research Areas:  

Cancer

AJICAP reagent 6b is an Fc-affinity peptide reagent that site-specifically modifies Lys288 of native antibodies via thiophenyl ester chemistry. AJICAP reagent 6b enables site-specific conjugation of native antibodies at Lys288 with high conversion yield and reduced aggregation. AJICAP reagent 6b can be used for the research of cancer .
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