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Cat. No.: HY-120223

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BMS-196085

BMS-196085 is an orally active, potent and selective full agonist against human β₃ adrenergic receptor with a K_i value of 21 nM. BMS-196085 also has partial agonist activity at the β₁ receptor. BMS-196085 is promising for research of obesity and type-II diabetes.

For research use only. We do not sell to patients.

CAS No.: 170686-10-9
Formula: C₂₄H₂₆F₂N₂O₅S
Molecular Weight:492.54

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (270 KB)

BMS-196085 Chemical Structure

CAS No.: 170686-10-9

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Use of MCE Products

Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

All Adrenergic Receptor Isoforms :

Chemical Information

CAS No. 170686-10-9
Molecular Weight 492.54
Formula C₂₄H₂₆F₂N₂O₅S
SMILES

O[C@H](C1=CC(NS(C)(=O)=O)=C(C=C1)O)CN[C@@H](C2=CC=C(C=C2)OC(F)F)CC3=CC=CC=C3
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (270 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Gavai A V, et al. BMS-196085: a potent and selective full agonist of the human β3 adrenergic receptor[J]. Bioorganic & medicinal chemistry letters, 2001, 11(23): 3041-3044.

[2]. Hu B, et al. Orally bioavailable β3-adrenergic receptor agonists as potential therapeutic agents for obesityand type-II diabetes[J]. Progress in medicinal chemistry, 2003, 41: 167-194.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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BMS-196085

All Adrenergic Receptor Isoforms

Biological Activity

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

BMS-196085 Related Classifications

HY-120223 Related Classifications