α2C adrenoceptor agonist 1
α2C adrenoceptor agonist 1 (Compound A) is an orally active, highly selective, and non-central nervous system penetrating agonist for the α2C-adrenoceptor, with EC50 and Ki values of 108 nM and 12 nM, respectively. α2C adrenoceptor agonist 1 can be used in the study of nasal congestion.
For research use only. We do not sell to patients.
- CAS No.: 928115-79-1
- Formula: C16H21N5O2
- Molecular Weight:315.37
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Adrenergic Receptor Isoforms
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Biological Activity
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Alpha-2C adrenergic receptor 108 nM (EC50) |
Alpha-2C adrenergic receptor 12 nM (Ki) |
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 928115-79-1
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Molecular Weight 315.37
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Formula C16H21N5O2
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SMILES
O=C(N(CC)C1=CC=C2OCCN(CC3=CN=CN3)C2=C1)NC
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)