1. GPCR/G Protein
  2. GNRH Receptor

Cetrorelix Acetate (Synonyms: SB-075 acetate; NS-75A)

Cat. No.: HY-P0009A Purity: 98.88%
Handling Instructions

Cetrorelix Acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with IC50 of 1.21 nM.

For research use only. We do not sell to patients.
Cetrorelix Acetate Chemical Structure

Cetrorelix Acetate Chemical Structure

CAS No. : 145672-81-7

Size Price Stock Quantity
1 mg USD 60 In-stock
5 mg USD 108 In-stock
10 mg USD 180 In-stock
25 mg USD 372 In-stock
50 mg USD 612 In-stock
100 mg   Get quote  
200 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Protocol

  • Technical Information

  • Purity & Documentation

  • References

Description

Cetrorelix Acetate is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with IC50 of 1.21 nM. target: GnRH [3] IC50: 1.21 nM [3] In vitro: GnRH-I antagonist Cetrorelix inhibit growth of ES-2 cell line only at 1000 ng/ml. [1] In vivo: Cetrorelix Exhibits antiproliferative effects and displays efficacy against hormone-sensitive cancers. Cetrorelix fully blocks the impairment of the consolidation of passive avoidance learning Cetrorelix elicit anxiolytic action and antidepressive-like action. Suppresses production of luteinizing hormone (LH) and follicle-stimulating hormone (FSH) from the pituitary gland lead to inhibit ovulation. [2]

Clinical Trial
References
Molecular Weight

1491.09

Formula

C₇₂H₉₆ClN₁₇O₁₆

CAS No.

145672-81-7

SMILES

[AFASYXLRPA acetate]

Storage
Protect from light
Powder -80°C 2 years
  -20°C 1 year
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

H2O: 5 mg/mL (Need ultrasonic)

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

Inquiry Online

Your information is safe with us. * Required Fields.

Product name

 

Salutation

Applicant name *

 

Email address *

Phone number *

 

Organization name *

Country *

 

Requested quantity *

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
Cetrorelix Acetate
Cat. No.:
HY-P0009A
Quantity: