1. Membrane Transporter/Ion Channel
  2. Sodium Channel

PF 04531083 

Cat. No.: HY-105283
Handling Instructions

PF 04531083 is a selective NaV1.8 blocker, and used for the research of neuropathic/inflammatory pain.

For research use only. We do not sell to patients.

PF 04531083 Chemical Structure

PF 04531083 Chemical Structure

CAS No. : 1079400-07-9

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  • Technical Information

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Description

PF 04531083 is a selective NaV1.8 blocker, and used for the research of neuropathic/inflammatory pain.

IC50 & Target

NaV1.8[1]

Clinical Trial
Solvent & Solubility
In Vitro: 

10 mM in DMSO

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.7949 mL 13.9747 mL 27.9494 mL
5 mM 0.5590 mL 2.7949 mL 5.5899 mL
10 mM 0.2795 mL 1.3975 mL 2.7949 mL
*Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

357.79

Formula

C₁₇H₁₆ClN₅O₂

CAS No.

1079400-07-9

SMILES

ClC1=CC=C(OC)C=C1C2=C(N=C(NC(C3=CC=NN3C)=O)C=C2)N

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

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Product Name:
PF 04531083
Cat. No.:
HY-105283
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PF 04531083

Cat. No.: HY-105283