1. Signaling Pathways
  2. Apoptosis
  3. PKD
  4. PKD Inhibitors

PKD Inhibitors

PKD1

PKD2

PKD3

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PKD Inhibitors
Product Name PKD1 PKD2 PKD3 Purity
CRT0066101 dihydrochloride
PKD1, IC50: 1 nM
PKD2, IC50: 2.5 nM
PKD3, IC50: 2 nM
99.92%
1-Naphthyl PP1
PKD1, IC50: 154.6 nM
PKD2, IC50: 133.4 nM
PKD3, IC50: 109.4 nM
99.08%
CID755673
PKD1, IC50: 182 nM
PKD2, IC50: 280 nM
PKD3, IC50: 227 nM
99.12%
CRT0066101
PKD1, IC50: 1 nM
PKD2, IC50: 2.5 nM
PKD3, IC50: 2 nM
kb NB 142-70
PKD1, IC50: 28.3 nM
PKD2, IC50: 58.7 nM
PKD3, IC50: 53.2 nM
98.08%
3-IN-PP1
PKD1, IC50: 108 nM
Cellular PKD2, IC50: 94 nM
PKD3, IC50: 108 nM
BPKDi
PKD1, IC50: 1 nM
PKD2, IC50: 9 nM
PKD3, IC50: 1 nM
≥99.0%
Protein kinase D inhibitor 1
PKD1, IC50: 35 ± 10 nM
PKD2, IC50: 35 ± 5 nM
PKD3, IC50: 17 ± 8 nM