1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
  3. GLUT
  4. GLUT Inhibitors

GLUT Inhibitors

GLUT1

GLUT2

GLUT3

GLUT4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

GLUT Inhibitors, Activators, Modulators & Substrates
Product Name GLUT1 GLUT2 GLUT3 GLUT4 Purity
BAY-876
GLUT1, IC50: 2 nM
GLUT2, IC50: 10.08 μM
GLUT3, IC50: 1.67 μM
GLUT4, IC50: 0.29 μM
99.67%
Phloretin
GLUT1
GLUT2
    99.92%
WZB117
GLUT1
      99.93%
KL-11743
GLUT1, IC50: 115 nM
GLUT2, IC50: 137 nM
GLUT3, IC50: 90 nM
GLUT4, IC50: 68 nM
99.40%
FKL-137
GLUT1
     
HK2-IN-3
GLUT1
   
GLUT4
(-)-Epicatechin gallate
GLUT1
      99.96%
Rhoifolin      
GLUT4
99.25%
STF-31
GLUT1, IC50: 1 μM
      99.79%
MOTS-c (human)      
GLUT4
99.90%
MOTS-c(human) acetate      
GLUT4
99.74%
D927      
GLUT4, EC50: 0.14 μM
99.46%
GLUT inhibitor-1
GLUT1, IC50: 242 nM
 
GLUT3, IC50: 179 nM
  99.03%
Avicularin      
GLUT4
99.80%
Fasentin      
GLUT4, IC50: 68 μM
98.0%
GLUT4-IN-2
GLUT1, IC50: 11.4 μM
   
GLUT4, IC50: 6.8 μM
99.17%
Zingibroside R1
GLUT1
      99.75%
Licarin B      
GLUT4
99.93%
Hydroxylamine (50% w/w in water)
GLUT1
     
Allyl methyl sulfide  
GLUT2
    98.0%
4'-Bromo-resveratrol
GLUT1
      99.94%
DS02312223      
GLUT4
98.24%
NGI-235
GLUT1
      99.70%
2-Amino-2-deoxyglucose hydrochloride
GLUT1
      98.0%
Deoxyandrographolide      
GLUT4
98.0%
Sennidin B      
GLUT4
99.25%
Cichoriin      
GLUT4
99.9%
Pterosin A      
GLUT4
Lavendustin B
GLUT1, Ki: 15 μM
      98.02%
4,6-O-Ethylidene-α-D-glucose
GLUT1
      98.0%
Phloretin (Standard)
GLUT1
GLUT2
   
GLUT1/EGFR-IN-1
GLUT1
      99.75%
Hypoglycemic agent 4  
GLUT2
   
GLUT1-IN-1
GLUT1
     
3-Fluoro-evodiamine glucose
GLUT1
     
Allyl methyl sulfide (Standard)  
GLUT2
   
CDr17
GLUT1
     
BR103354
GLUT1
     
NIR‐fluorescent glucose  
GLUT2
 
GLUT4
DS-1150b      
GLUT4
Hydrangeic acid      
GLUT4
NV-5440
GLUT1
GLUT2
GLUT3
GLUT4
Avicularin (Standard)      
GLUT4
GLUT4 activator 3      
GLUT4
(Rac)-Glutipyran
GLUT1
 
GLUT3
 
Antidiabetic agent 7      
GLUT4
Sennidin A      
GLUT4