2. Membrane Transporter/Ion Channel
  3. EHD Protein ATP Synthase
  4. ATPase-IN-4

ATPase-IN-4 (Compound MS1) inhibits the ATPase activity of EHD4 (IC50: 0.92 μM). ATPase-IN-4 also inhibits EHD2 enzymatic activity

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ATPase-IN-4

ATPase-IN-4 Chemical Structure

CAS No. : 1219577-48-6

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Based on 1 publication(s) in Google Scholar

ATPase-IN-4 Related Antibodies

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Description

ATPase-IN-4 (Compound MS1) inhibits the ATPase activity of EHD4 (IC50: 0.92 μM). ATPase-IN-4 also inhibits EHD2 enzymatic activity[1]

IC50 & Target

EHD2

 

Molecular Weight

356.44

Formula

C19H20N2O3S
CAS No.
Appearance

Solid

Color

Light yellow to brown

SMILES

O=C(NC1=CC=CC=C1O)CCCCCN2SC3=CC=CC=C3C2=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (280.55 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.8055 mL 14.0276 mL 28.0552 mL
5 mM 0.5611 mL 2.8055 mL 5.6110 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass
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Concentration
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Volume
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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start)

C1

×
Volume (start)

V1

=
Concentration (final)

C2

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Volume (final)

V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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g

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(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 98.25%

SDS (251 KB)

COA (246 KB) HNMR (268 KB) LCMS (97 KB)

Handling Instructions (2659 KB)
References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.8055 mL 14.0276 mL 28.0552 mL 70.1380 mL
5 mM 0.5611 mL 2.8055 mL 5.6110 mL 14.0276 mL
10 mM 0.2806 mL 1.4028 mL 2.8055 mL 7.0138 mL
15 mM 0.1870 mL 0.9352 mL 1.8703 mL 4.6759 mL
20 mM 0.1403 mL 0.7014 mL 1.4028 mL 3.5069 mL
25 mM 0.1122 mL 0.5611 mL 1.1222 mL 2.8055 mL
30 mM 0.0935 mL 0.4676 mL 0.9352 mL 2.3379 mL
40 mM 0.0701 mL 0.3507 mL 0.7014 mL 1.7535 mL
50 mM 0.0561 mL 0.2806 mL 0.5611 mL 1.4028 mL
60 mM 0.0468 mL 0.2338 mL 0.4676 mL 1.1690 mL
80 mM 0.0351 mL 0.1753 mL 0.3507 mL 0.8767 mL
100 mM 0.0281 mL 0.1403 mL 0.2806 mL 0.7014 mL
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ATPase-IN-4 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

ATPase-IN-41219577-48-6EHD ProteinATP SynthaseEps15 Homology Domain (EHD) ProteinEHD proteinsATPase assayInhibitorinhibitorinhibit

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