BHEPN
BHEPN is an inhibitor of vascular endothelial growth factor receptor-2 (VEGFR-2). BHEPN has inhibition of VEGFR-2 with an IC50 value of 0.320 μM. BHEPN also exhibits remarkable cytotoxic effects against HepG2 and MCF-7 cancer cell lines, with IC50 values of 0.19 μM and 1.18 μM, respectively. BHEPN can be used for anticancer research.
For research use only. We do not sell to patients.
- Formula: C21H17BrN4O2
- Molecular Weight:437.29
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All VEGFR Isoforms
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Biological Activity
IC50: 0.320 μM (VEGFR-2); 0.19 μM (HepG2); 1.18 μM (MCF-7)[1]
Chemical Information
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Molecular Weight 437.29
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Formula C21H17BrN4O2
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SMILES
O=C(NC1=CC=CC(/C(C)=N/NC(C2=CC=C(Br)C=C2)=O)=C1)C3=CN=CC=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)