BQZ-485
BQZ-485 is a a potent GDI2 inhibitor through the interaction with Tyr245. BQZ-485 disrupts the intrinsic GDI2-Rab1A interaction, thereby abolishing vesicular transport from the endoplasmic reticulum (ER) to the Golgi apparatus and initiating subsequent paraptosis events.
For research use only. We do not sell to patients.
- CAS No.: 1906915-49-8
- Formula: C32H39NO3
- Molecular Weight:485.66
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
GDI2 |
Chemical Information
-
CAS No. 1906915-49-8
-
Molecular Weight 485.66
-
Formula C32H39NO3
-
SMILES
CC1=CC(C)=CC(COC2=CC3=C([C@](C[C@@H](O)C[C@@H]4C)([H])N4CC3)C=C2OCC5=CC(C)=CC(C)=C5)=C1
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)