AP-238
AP-238 is a a new synthetic opioid (NSO), and acts as an agonist for μ-opioid receptor (MOR) with an EC50 of 248 nM. AP-238 exhibits analgesic activity.
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- CAS No.: 140924-11-4
- Formule: C18H26N2O
- Masse moléculaire:286.41
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Description
IC50 & Target
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μ Opioid Receptor/MOR 248 nM (EC50) |
Chemical Information
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CAS No. 140924-11-4
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Masse moléculaire 286.41
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Formule C18H26N2O
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SMILES
CCC(N1[C@H](C)CN(C/C=C/C2=CC=CC=C2)C[C@@H]1C)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
[1]. Jurowski K, et, al. Prediction of key toxicity endpoints of AP-238 a new psychoactive substance for clinical toxicology and forensic purposes using in silico methods. Sci Rep. 2024 Nov 22;14(1):28977. [Content Brief]
[2]. Brunetti P, et al., Human metabolism and basic pharmacokinetic evaluation of AP-238: A recently emerged acylpiperazine opioid. Drug Test Anal. 2024 Feb;16(2):221-235. [Content Brief]
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
AP-238 Related Classifications
HY-170310 Related Classifications
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