R-84760
R-84760 is a selective κ-opioid receptor agonist. R-84760 has antinociceptive effect.
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- CAS No.: 157824-23-2
- Formule: C19H25Cl3N2OS
- Masse moléculaire:435.84
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
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Activité biologique
Description
IC50 & Target
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κ Opioid Receptor/KOR |
In Vitro
In an opioid receptor binding assay with a guinea pig brain membrane fraction, R-84760 shows a 5 times higher affinity for the kappa-opioid receptor than CI-977 (HY-105235). The selectivity of R-84760 for the kappa-opioid receptor is higher than that of U-69593 (HY-12363)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 157824-23-2
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Masse moléculaire 435.84
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Formule C19H25Cl3N2OS
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SMILES
O=C([C@H]1CCC2=C1C=C(Cl)C(Cl)=C2)N3[C@H](CN4CCCC4)CSCC3.Cl
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
R-84760 Related Classifications
HY-19206 Related Classifications
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