1104662-66-9
Chemical Structure
SNT-207858 free base
- CAS No.: 1104662-66-9
- Formula:C32H43Cl2N5O3
- Molecular Weight:616.62
IUPAC Name: N-((R)-3-(2,4-dichlorophenyl)-1-oxo-1-(4-(3-((R)-2-(pyrrolidin-1-yl)butoxy)pyridin-2-yl)piperidin-1-yl)propan-2-yl)pyrrolidine-1-carboxamide
InChIKey: GNSVFEJLUPMLCZ-IXCJQBJRSA-N
SMILES: O=C(N1CCCC1)N[C@H](CC2=CC=C(Cl)C=C2Cl)C(N3CCC(C4=NC=CC=C4OC[C@H](N5CCCC5)CC)CC3)=O
Biological Activity: SNT207858 free base is a selective, blood brain barrier penetrating, potent and orally active melanocortin-4 (MC-4) receptor antagonist. SNT207858 free base has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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SNT-207858 free base | 99.66% | SNT207858 free base is a selective, blood brain barrier penetrating, potent and orally active melanocortin-4 (MC-4) receptor antagonist. SNT207858 free base has an IC50 of 22 nM (binding) and 11 nM (function) on the MC-4 receptor. | ||||||||||||||||||||
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Keywords
