136647-02-4
136647-02-4
Chemical Structure
UK-78282 hydrochloride
- CAS No.: 136647-02-4
- Formula:C29H36ClNO2
- Molecular Weight:466.05
IUPAC Name: 4-((benzhydryloxy)methyl)-1-(3-(4-methoxyphenyl)propyl)piperidine hydrochloride
InChIKey: ZZSQARULZYQMIG-UHFFFAOYSA-N
SMILES: COC1=CC=C(CCCN2CCC(COC(C3=CC=CC=C3)C4=CC=CC=C4)CC2)C=C1.[H]Cl
Biological Activity: UK-78282, a novel piperidine, potent and selective Kv1.3 blocker with an IC50 of 200 nM. UK-78,282 effectively suppresses human T-lymphocyte activation in vitro. UK-78,282 binds to residues at the inner surface of the channel overlapping the site of action of verapamil[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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UK-78282 hydrochloride | 99.82% | UK-78282, a novel piperidine, potent and selective Kv1.3 blocker with an IC50 of 200 nM. UK-78,282 effectively suppresses human T-lymphocyte activation in vitro. UK-78,282 binds to residues at the inner surface of the channel overlapping the site of action of verapamil. | ||||||||||||||||||||
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References
Keywords
