191672-52-3
Chemical Structure
CS-003 Free base
- CAS 番号: 191672-52-3
- Formula:C34H38Cl2N2O6S
- Molecular Weight:673.65
IUPAC Name: ((R)-2-(3,4-dichlorophenyl)-2-(2-((S)-2-oxido-3H-spiro[benzo[c]thiophene-1,4'-piperidin]-1'-yl)ethyl)morpholino)(3,4,5-trimethoxyphenyl)methanone
InChIKey: RWSBBXFLRGQFQP-RKCQUONGSA-N
SMILES: O=C(N1C[C@@](CCN2CCC3(CC2)C4=CC=CC=C4C[S@@]3=O)(C5=CC=C(Cl)C(Cl)=C5)OCC1)C6=CC(OC)=C(OC)C(OC)=C6
Biological Activity: CS-003 Free base (CS-003), a triple tachykinin receptor antagonist, shows high affinities for human (Neurokinin) NK1, NK2 and NK3 receptors with Ki values of 2.3 nM, 0.54 nM and 0.74 nM, respectively. CS-003 Free base (CS-003) has therapeutic efficacy on respiratory diseases associated with neurokinins.
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CS-003 Free base | CS-003 Free base (CS-003), a triple tachykinin receptor antagonist, shows high affinities for human (Neurokinin) NK1, NK2 and NK3 receptors with Ki values of 2.3 nM, 0.54 nM and 0.74 nM, respectively. CS-003 Free base (CS-003) has therapeutic efficacy on respiratory diseases associated with neurokinins. | |||||||||||||||||||||
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