2225800-19-9
2225800-19-9
Chemical Structure
PARP10-IN-3
- No. CAS: 2225800-19-9
- Formula:C14H12N2O3
- Molecular Weight:256.26
IUPAC Name: 3-(4-carbamoylphenoxy)benzamide
InChIKey: PMOXYDXLQIUWHL-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(C=C1)OC2=CC=CC(C(N)=O)=C2)N
Biological Activity: PARP10-IN-3 is a selective mono‐ADP‐ribosyltransferase PARP10 inhibitor with an IC50 of 480 nM for human PARP10. PARP10-IN-3 reveals potent inhibition on PARP2 and PARP15 with IC50s of 1.7 μM for human PARP2 and human PARP15, respectively[1].
| Referencia número | Nombre del producto | Pureza | Descripciòn | Pricing | |||||||||||||||||||
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PARP10-IN-3 | 98.72% | PARP10-IN-3 is a selective mono‐ADP‐ribosyltransferase PARP10 inhibitor with an IC50 of 480 nM for human PARP10. PARP10-IN-3 reveals potent inhibition on PARP2 and PARP15 with IC50s of 1.7 μM for human PARP2 and human PARP15, respectively. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 0.87
HY-123512OUL35 -
Similarity Score 0.77
HY-148753PARP10-IN-2 -
Similarity Score 0.77
HY-W340326(4′-Hydroxy)phenoxybenzoic acid -
Similarity Score 0.75
HY-W0118254,4'-Oxybis(benzoic acid) -
Similarity Score 0.75
HY-445904,4'-Oxydibenzoyl chloride -
Similarity Score 0.72
HY-788544-Phenoxybenzoic acid -
Similarity Score 0.72
HY-W014225R3-Phenoxybenzoic acid (Standard) -
Similarity Score 0.72
HY-W014225S3-Phenoxybenzoic acid-13C6 -
Similarity Score 0.71
HY-118615LY2048978 -
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