2307461-45-4
Chemical Structure
FAK ligand-Linker Conjugate 1
- CAS No.: 2307461-45-4
- Formula:C25H28F3N5O6S
- Molecular Weight:583.58
IUPAC Name: 3-(2-(4-((4-((3-(N-methylmethylsulfonamido)benzyl)amino)-5-(trifluoromethyl)pyrimidin-2-yl)amino)phenoxy)ethoxy)propanoic acid
InChIKey: OSVHAJNGZCDBGV-UHFFFAOYSA-N
SMILES: O=C(O)CCOCCOC1=CC=C(NC2=NC=C(C(F)(F)F)C(NCC3=CC=CC(N(C)S(=O)(C)=O)=C3)=N2)C=C1
Biological Activity: FAK ligand-Linker Conjugate 1 incorporates a ligand for FAK, and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). FAK ligand-Linker Conjugate 1 can be extensively used for PROTAC-mediated protein degradation[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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FAK ligand-Linker Conjugate 1 | 98.91% | FAK ligand-Linker Conjugate 1 incorporates a ligand for FAK, and a PROTAC linker, which recruit E3 ligases (such as VHL, CRBN, MDM2, and IAP). FAK ligand-Linker Conjugate 1 can be extensively used for PROTAC-mediated protein degradation. | ||||||||||||||||||||
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Keywords
