2492596-61-7
2492596-61-7
Chemical Structure
MRGPRX4 modulator-1
- CAS No.: 2492596-61-7
- Formula:C16H13ClF3NO3
- Molecular Weight:359.73
IUPAC Name: 6-((2-chloro-4-(trifluoromethyl)phenoxy)methyl)-4-ethylpicolinic acid
InChIKey: UNHAKUSQBBXQSU-UHFFFAOYSA-N
SMILES: O=C(C1=NC(COC2=CC=C(C(F)(F)F)C=C2Cl)=CC(CC)=C1)O
Biological Activity: MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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MRGPRX4 modulator-1 | 98.13% | MRGPRX4 modulator-1 (compound 31-2) is a potent mas-related g-protein receptor X4 (MRGPR X4) modulator, with antagonist activity of IC50 < 100 nM for MRGPR4. MRGPRX4 modulator-1 can be used for researching MRGPR X4 dependent diseases such as itch, pain, and autoimmune disorders. | ||||||||||||||||||||
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Structural Analogs
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HY-147051Nelremagpran -
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HY-160002MAO-B-IN-27 -
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HY-138997MBX-102 acid -
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HY-W4565215-((4-Carboxyphenoxy)methyl)isophthalic acid -
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HY-108494CYM50260 -
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HY-W5869344-(3-Carboxyphenyl)-2,6-pyridinedicarboxylic acid -
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