2930378-91-7
2930378-91-7
Chemical Structure
GAK inhibitor 49 hydrochloride
- CAS. Nr.: 2930378-91-7
- Formula:C20H23ClN2O5
- Molecular Weight:406.86
IUPAC Name: 6,7-dimethoxy-N-(3,4,5-trimethoxyphenyl)quinolin-4-amine hydrochloride
InChIKey: LOOMZTXOCDWFDB-UHFFFAOYSA-N
SMILES: COC1=C(OC)C(OC)=CC(NC2=CC=NC3=CC(OC)=C(OC)C=C23)=C1.[H]Cl
Biological Activity: GAK inhibitor 49 hydrochloride is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 hydrochloride also shows binding to RIPK2[1].
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GAK inhibitor 49 hydrochloride | 99.52% | GAK inhibitor 49 hydrochloride is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. GAK inhibitor 49 hydrochloride also shows binding to RIPK2. | ||||||||||||||||||||
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