824982-41-4
Chemical Structure
A-784168
- CAS No.: 824982-41-4
- Formula:C19H15F6N3O3S
- Molecular Weight:479.40
IUPAC Name: 3'-(trifluoromethyl)-N-(4-((trifluoromethyl)sulfonyl)phenyl)-3,6-dihydro-2H-[1,2'-bipyridine]-4-carboxamide
InChIKey: SDUAWRFBHRAFBM-UHFFFAOYSA-N
SMILES: O=C(C1=CCN(C2=NC=CC=C2C(F)(F)F)CC1)NC3=CC=C(S(=O)(C(F)(F)F)=O)C=C3
Biological Activity: A-784168 is a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1). Vanilloid receptor type 1 (TRPV1) is a ligand-gated nonselective cation channel that is considered to be an important integrator of various pain stimuli such as endogenous lipids, capsaicin, heat, and low pH. A-784168 has good CNS penetration[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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A-784168 | 99.79% | A-784168 is a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1). Vanilloid receptor type 1 (TRPV1) is a ligand-gated nonselective cation channel that is considered to be an important integrator of various pain stimuli such as endogenous lipids, capsaicin, heat, and low pH. A-784168 has good CNS penetration. | ||||||||||||||||||||
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A-784168 (Standard) | ≥98% | A-784168 (Standard) is the analytical standard of A-784168 (HY-108460). This product is intended for research and analytical applications. A-784168 is a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1). Vanilloid receptor type 1 (TRPV1) is a ligand-gated nonselective cation channel that is considered to be an important integrator of various pain stimuli such as endogenous lipids, capsaicin, heat, and low pH. A-784168 has good CNS penetration. | ||||||||||||||||||||
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