83397-56-2
83397-56-2
Chemical Structure
PL-017
- CAS No.: 83397-56-2
- Formula:C29H37N5O5
- Molecular Weight:535.63
IUPAC Name: (S)-1-(L-tyrosyl)-N-((S)-1-((R)-2-carbamoylpyrrolidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-N-methylpyrrolidine-2-carboxamide
InChIKey: JAKBYSTWCHUQOK-NDBXHCKUSA-N
SMILES: O=C(N1[C@H](CCC1)C(N)=O)[C@H](CC2=CC=CC=C2)N(C)C([C@H]3N(CCC3)C([C@@H](N)CC4=CC=C(O)C=C4)=O)=O
Biological Activity: PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats[1].
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PL-017 | PL-017 is a potent and selective μ opioid receptor agonist with an IC50 of 5.5 nM for 125I-FK 33,824 binding to μ site. PL-017 produces long-lasting, reversible analgesia in rats. | |||||||||||||||||||||
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References
Keywords
