853260-98-7
853260-98-7
Chemical Structure
GPR109 receptor agonist-4
- CAS No.: 853260-98-7
- Formula:C13H12O4
- Molecular Weight:232.23
InChIKey: SUHZZFNDVLWPTL-UHFFFAOYSA-N
SMILES: O=C(C(OC1(CC)C2=CC=CC=C2)=CC1=O)O
Biological Activity: GPR109 receptor agonist-4 is a high-affinity GPR109a and low-affinity GPR109b niacin receptor agonist with EC50 values of 24 μM and 4.8 μM, respectively. GPR109 receptor agonist-4 acts through Gi-coupled receptors to reduce intracellular cAMP, which in turn negatively regulates hormone-sensitive lipase activity and inhibits lipolysis. GPR109 receptor agonist-4 can be used in the study of atherosclerosis[1].
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GPR109 receptor agonist-4 | GPR109 receptor agonist-4 is a high-affinity GPR109a and low-affinity GPR109b niacin receptor agonist with EC50 values of 24 μM and 4.8 μM, respectively. GPR109 receptor agonist-4 acts through Gi-coupled receptors to reduce intracellular cAMP, which in turn negatively regulates hormone-sensitive lipase activity and inhibits lipolysis. GPR109 receptor agonist-4 can be used in the study of atherosclerosis. | |||||||||||||||||||||
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