893428-72-3
893428-72-3
Chemical Structure
Saracatinib difumarate
Synonym(s): AZD0530 difumarate
- CAS No.: 893428-72-3
- Formula:C35H40ClN5O13
- Molecular Weight:774.17
IUPAC Name: N-(5-chlorobenzo[d][1,3]dioxol-4-yl)-7-(2-(4-methylpiperazin-1-yl)ethoxy)-5-((tetrahydro-2H-pyran-4-yl)oxy)quinazolin-4-amine difumarate
InChIKey: OQXMMAQEMJUIQM-LVEZLNDCSA-N
SMILES: ClC1=CC=C2C(OCO2)=C1NC3=C4C(OC5CCOCC5)=CC(OCCN6CCN(C)CC6)=CC4=NC=N3.OC(/C=C/C(O)=O)=O.OC(/C=C/C(O)=O)=O
Biological Activity: Saracatinib (AZD0530) difumarate is a potent Src inhibitor with IC50 values of 2.7-11 nM for c-Src, Lck, c-YES, Lyn, Fyn, Fgr and Blk, and is selective for other tyrosine kinases. [1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Saracatinib difumarate | 99.93% | Saracatinib (AZD0530) difumarate is a potent Src inhibitor with IC50 values of 2.7-11 nM for c-Src, Lck, c-YES, Lyn, Fyn, Fgr and Blk, and is selective for other tyrosine kinases. . | ||||||||||||||||||||
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Saracatinib difumarate (Standard) | ≥98% | Saracatinib (difumarate) (Standard) is the analytical standard of Saracatinib (difumarate). This product is intended for research and analytical applications. Saracatinib (AZD0530) difumarate is a potent Src inhibitor with IC50 values of 2.7-11 nM for c-Src, Lck, c-YES, Lyn, Fyn, Fgr and Blk, and is selective for other tyrosine kinases. . | ||||||||||||||||||||
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References
