CaSR antagonist-1
CaSR antagonist-1 is a calcium sensing receptor (CaSR) antagonist with an IC50 value of 50 nM. CaSR antagonist-1 can be used for the research of disorders associated with abnormal bone or mineral homeostasis such as osteoporosis.
For research use only. We do not sell to patients.
- CAS No.: 1219811-83-2
- Formula: C29H24FN3O2S
- Molecular Weight:497.58
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
IC50:50 nM (CaSR)[1].EC50:＞50 μM (hPXR Gene reporter assay)[1].
Chemical Information
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CAS No. 1219811-83-2
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Molecular Weight 497.58
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Formula C29H24FN3O2S
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SMILES
O=C1C(C2=CC(C3=CC=CC=N3)=C(C)S2)=C(C)N=C(N1CCC4=CC=CC=C4)C5=C(O)C(F)=CC=C5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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