1. Membrane Transporter/Ion Channel
    Neuronal Signaling
  2. GABA Receptor
  3. CGP 36742

CGP 36742 (Synonyms: SGS-742)

Cat. No.: HY-121599 Purity: >97.0%
Handling Instructions

CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood–brain barrier after peripheral administration, with an IC50 of 32 μM. CGP 36742 is useful in treatment of depression.

For research use only. We do not sell to patients.

CGP 36742 Chemical Structure

CGP 36742 Chemical Structure

CAS No. : 123690-78-8

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1 mg USD 90 In-stock
Estimated Time of Arrival: December 31
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Based on 1 publication(s) in Google Scholar

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Description

CGP 36742 is a selective GABAB receptor antagonist that can penetrate the blood–brain barrier after peripheral administration, with an IC50 of 32 μM. CGP 36742 is useful in treatment of depression[1].

IC50 & Target

IC50: 32 μM (GABAB)[1]

Molecular Weight

179.20

Formula

C₇H₁₈NO₂P

CAS No.

123690-78-8

SMILES

O=P(CCCN)(O)CCCC

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Pure form -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References

Purity: >97.0%

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CGP 36742
Cat. No.:
HY-121599
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