CK2-IN-3
CK2-IN-3 is a selective and potent CK2 inhibitor (Kd: 12 nM), with IC50 values of 1.51 μM (CK2α) and 7.64 μM (CK2α’). CK2-IN-3 can be used in the research of cancers.
For research use only. We do not sell to patients.
- CAS No.: 2969205-85-2
- Formula: C22H26N4O7
- Molecular Weight:458.46
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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CK2α 1.51 μM (IC50) |
CK2α' 7.64 μM (IC50) |
CK2-IN-3 (compound 31, 1 nM-100 μM) inhibits CK2 activities in permeabilized cells, with IC50 values of 8 nM (CK2α) and 38 nM (CK2α’)[1].
CK2-IN-3 (10 µM, 48 h) shows no significant cytotoxicity across 60 cancer cell lines[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2969205-85-2
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Molecular Weight 458.46
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Formula C22H26N4O7
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SMILES
O=C(O)C1=CC=C(C2=C3N=C(N(C(OC(C)(C)C)=O)CCOCCO)C=CN3N=C2)C=C1O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CK2-IN-3 Related Classifications
HY-151382 Related Classifications
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