1410101-89-1
1410101-89-1
Chemical Structure
(R)-PS210
- CAS No.: 1410101-89-1
- Formula:C19H15F3O5
- Molecular Weight:380.31
IUPAC Name: (R)-2-(3-oxo-1-phenyl-3-(4-(trifluoromethyl)phenyl)propyl)malonic acid
InChIKey: MLJPLHGJBUWCBA-AWEZNQCLSA-N
SMILES: O=C(O)C([C@H](C1=CC=CC=C1)CC(C2=CC=C(C(F)(F)F)C=C2)=O)C(O)=O
Biological Activity: (R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket of?PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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(R)-PS210 | 98.09% | (R)-PS210, the R enantiomer of PS210 (compound 4h-eutomer), is a substrate-selective allosteric activator of PDK1 with an AC50 value of 1.8 μM. (R)-PS210 targets to the PIF-binding pocket of?PDK1. PIF: The protein kinase C-related kinase 2 (PRK2)-interacting fragment. | ||||||||||||||||||||
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Structural Analogs
-
Similarity Score 1.00
HY-121629PS210 -
Similarity Score 0.71
HY-124060PS423 -
Similarity Score 0.60
HY-W10605711β-HSD1-IN-7 -
Similarity Score 0.56
HY-W628136MAO-B-IN-47 -
Similarity Score 0.55
HY-N11597Daphneolone -
Similarity Score 0.55
HY-116263CATPB -
Similarity Score 0.55
HY-W5437481,3,5-Triphenylpentane-1,5-dione -
Similarity Score 0.54
HY-B1138Fenbufen -
Similarity Score 0.54
HY-W000795(S)-2-amino-3-(4-benzoylphenyl)propanoic acid -
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