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Referencia número: HY-181584

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AKI-062a

AKI-062a is a non-selective kinase inhibitor, such as a CK1γ inhibitor. AKI-062a binds to and inhibits WNT pathway kinases and GSK3β. At a concentration of 1 μM, AKI-062a binds to 17 kinases, with a binding activity of <10% of that of the control group.

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No. CAS: 1093303-07-1
Fòrmula: C₂₀H₂₁N₇O
Peso molecular:375.43

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

AKI-062a Chemical Structure

No. CAS: 1093303-07-1

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

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Descripciòn

IC₅₀ & Target

GSK-3β

Ver todos los productos específicos de isoformas GSK-3 :

In Vitro

AKI-062a (1 μM) demonstrates non-selective kinase binding, interacting with 17 kinases including the WNT pathway kinase GSK3β^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

No. CAS 1093303-07-1
Peso molecular 375.43
Fòrmula C₂₀H₂₁N₇O
SMILES

CN(C)CC(NC1=NNC(C1=C2)=CC=C2C(N=N3)=CN3CC4=CC=CC=C4)=O
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Capener JL, et al. Development of a Chemical Probe to Enable Characterization of the Casein Kinase 1γ Subfamily. J Med Chem. 2026 Feb 12;69(3):2666-2684. [Content Brief]

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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AKI-062a

Ver todos los productos específicos de isoformas GSK-3

Actividad biológica

Chemical Information

Pureza y Documentación

Referencias

Calculators

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AKI-062a Related Classifications

HY-181584 Related Classifications