GHSR-1a agonist-1
GHSR-1a agonist-1 (Compound 4b) is an orally active agonist of the human growth hormone secretagogue receptor 1a (GHSR-1a), with an EC50 of 0.49 nM. GHSR-1a agonist-1 can effectively stimulate the release of endogenous growth hormone by activating GHSR-1a. GHSR-1a agonist-1 administered orally at a dose as low as 0.1 mg/kg can increase the body weight and body length of 4-week-old rats. GHSR-1a agonist-1 can be used in the research field of growth and development retardation in children.
For research use only. We do not sell to patients.
- CAS No.: 3060887-25-1
- Formula: C30H37N5O4
- Molecular Weight:531.65
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
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GHSR1a 0.49 nM (IC50) |
Chemical Information
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CAS No. 3060887-25-1
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Molecular Weight 531.65
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Formula C30H37N5O4
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SMILES
O=C(N(CCC1=NN(C2=O)C3CC3)C[C@]12CC4=CC=CC=C4)[C@@H](COCC5=CC=CC=C5)NC(C(N)(C)C)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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