GLP-1R agonist 45
GLP-1R agonist 45 is a full GLP-1R agonist with an EC50 of 2.20 nM. GLP-1R agonist 45 can be used in the research of type 2 diabetes and obesity.
For research use only. We do not sell to patients.
- CAS No.: 2428641-61-4
- Formula: C31H30FN5O4
- Molecular Weight:555.60
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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GLP-1 2.20 nM (EC50) |
GLP-1R agonist 45 (Compound 4a) (1 μM; 15 min) fully activates GLP-1R in transiently transfected HEK293 cells, with an EC50 of 2.20 nM, making it a potent full agonist of this receptor[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 2428641-61-4
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Molecular Weight 555.60
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Formula C31H30FN5O4
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SMILES
O=C(C1=CC=C2C(N(C[C@H]3OCC3)C(CN4CCN(C5=CC=CC(OCC6=CC=C(C#N)C=C6F)=C5)CC4)=N2)=C1)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)