Glutaminase-IN-4
Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor with an IC50 of 2.3 μM.
For research use only. We do not sell to patients.
- CAS No.: 1439390-05-2
- Formula: C23H22N6O2S2
- Molecular Weight:478.59
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 2.3 μM (Glutaminase)[1]
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| NCI-H1703 | GI50 |
0.794 μM
Compound: 8
|
Antiproliferative activity against human NCI-H1703 cells assessed as reduction in cell growth after 5 days by SYTOX green staining-based assay
Antiproliferative activity against human NCI-H1703 cells assessed as reduction in cell growth after 5 days by SYTOX green staining-based assay
|
[PMID: 31199640] |
Chemical Information
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CAS No. 1439390-05-2
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Molecular Weight 478.59
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Formula C23H22N6O2S2
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SMILES
O=C(NC1=NN=C(S1)CCCC2=NN=C(S2)NC(CC3=CC=CC=C3)=O)CC4=CC=CC=C4
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)