Glutaminase-IN-4
Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor with an IC50 of 2.3 μM.
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- CAS 番号: 1439390-05-2
- 分子式: C23H22N6O2S2
- 分子量:478.59
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
製品説明
IC50 & Target
IC50: 2.3 μM (Glutaminase)[1]
Cellular Effect
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| NCI-H1703 | GI50 |
0.794 μM
Compound: 8
|
Antiproliferative activity against human NCI-H1703 cells assessed as reduction in cell growth after 5 days by SYTOX green staining-based assay
Antiproliferative activity against human NCI-H1703 cells assessed as reduction in cell growth after 5 days by SYTOX green staining-based assay
|
[PMID: 31199640] |
化学情報
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CAS 番号 1439390-05-2
-
分子量 478.59
-
分子式 C23H22N6O2S2
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SMILES
O=C(NC1=NN=C(S1)CCCC2=NN=C(S2)NC(CC3=CC=CC=C3)=O)CC4=CC=CC=C4
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輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)