GPR6 inverse agonist 2
GPR6 inverse agonist 2 (Compound 575) is a selective GPR6 inverse agonist, with IC50 values of < 0.1 μM and 1~30 μM against GPR6 and GPR3, respectively. GPR6 inverse agonist 2 exhibits preliminary cardiac safety, with an IC50 of 21.71 μM for hERG. GPR6 inverse agonist 2 can be used in the research of movement disorders such as Parkinson's disease.
For research use only. We do not sell to patients.
- CAS No.: 3029155-57-2
- Formula: C27H31F2N7O2
- Molecular Weight:523.58
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
Chemical Information
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CAS No. 3029155-57-2
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Molecular Weight 523.58
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Formula C27H31F2N7O2
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SMILES
CC(C)(O)[C@@H](O)C1=CC2=NC(N3CCN(CC4=CC=C(F)C=C4F)CC3)=C(C5=CN(CC)N=C5)N=C2C=N1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)