GSK-1562590
GSK-1562590 is a uropeptide-II receptor antagonist with high affinity and selectivity. GSK-1562590 exhibits significant antagonistic activity in multiple bioassays and, in contrast, displays relatively sustained receptor binding times. GSK-1562590 can inhibit human urinary peptide-II-induced aortic contraction in rats in experiments, and its effect can last for at least 24 hours.
For research use only. We do not sell to patients.
- CAS No.: 1003877-55-1
- Formula: C30H30Cl2N4O4
- Molecular Weight:581.49
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All Endogenous Metabolite Isoforms
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Biological Activity
Chemical Information
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CAS No. 1003877-55-1
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Molecular Weight 581.49
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Formula C30H30Cl2N4O4
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SMILES
NC(C1=CC=CC(C(C=C2)=CC=C2[C@H](CN3CCCC3)N(C)C(CN4C5=CC(Cl)=C(Cl)C=C5OCC4=O)=O)=C1)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)